反应条件
1: 1.) NaH, 3.) aq. NH3 / 1) DMF, 15 min; 2) DMF, 30 min; 3) overnight, room temperature
2: 1.) K2CO3 / 1) DMF, 30 min; 2) DMF, 45 min
3: 1.) N-bromosuccinimide, 2.) aq. NH3 / 1) water, 25 min; 2) room temperature, 30 min
View Scheme
参考文献
Boryski, Jerzy; Golankiewicz, Bozenna; Clercq, Erik De
Journal of Medicinal Chemistry, 1988 , vol. 31, # 7 p. 1351 - 1355
