2-(溴甲基)-5-氯噻吩合成路线 (共 2 条)
反应条件
phosphorus tribromide in diethyl ether
T=0 - 20°C; 48 h;
参考文献
PORTOLA PHARMACEUTICALS, INC.
Patent: WO2008/36843 A2, 2008 ;
Location in patent: Page/Page column 34 ;
WO 2008/036843 A2
参考文献
ELI LILLY AND COMPANY
Patent: WO2007/2181 A2, 2007 ;
Location in patent: Page/Page column 137 ;
WO 2007/002181 A2