反应条件
1: 1.) MeI, potassium carbonate / 1.) CH3CN, 5 deg C, 30 min, 2.) CH3CN, reflux, 15 h
2: conc. aq. HCl / 15 h / Heating
3: 76 percent / NH4OAc / acetic acid / 2 h / Heating
View Scheme
参考文献
Owton; Gallagher; Brunavs
Synthetic Communications, 1992 , vol. 22, # 3 p. 351 - 357