2-乙酰氨基-3-(4-联苯)丙烯酸合成路线 (共 2 条)
反应条件
water in acetone
8 h; Reflux;
参考文献
ZHEJIANG JIUZHOU PHARMACEUTICAL CO., LTD.; NOVARTIS AG; ZHU, Guoliang; SHI, Desong; WEI, Junhui; TAO, Fengfeng
Patent: WO2010/34236 A1, 2010 ;
Location in patent: Page/Page column 13 ;
WO 2010/034236 A1
反应条件
1: acetic anhydride; sodium acetate / 0.5 h / Reflux
2: water / acetone / 8 h / Reflux
View Scheme
参考文献
ZHEJIANG JIUZHOU PHARMACEUTICAL CO., LTD.; NOVARTIS AG; ZHU, Guoliang; SHI, Desong; WEI, Junhui; TAO, Fengfeng
Patent: WO2011/35569 A1, 2011 ;
WO 2011/035569 A1