1: With potassium permanganate in tetrahydrofuran T=20°C; 48 h; 2: With potassium hydroxide in tetrahydrofuran; water T=20°C; 2 h; 3: With hydrogenchloride in water
参考文献
AVIGEN, INC.
Patent: WO2007/146087 A2, 2007 ;
Location in patent: Page/Page column 75 ;
1: N,N-dimethyl-formamide With trichlorophosphate
T=20°C; 0.166667 h;
2: 2-isopropyl-pyrazolo[1,5-a]pyridine T=20°C; 19 h;
3: With sodium hydroxide in water
pH=8;
参考文献
AVIGEN, INC.
Patent: WO2007/146087 A2, 2007 ;
Location in patent: Page/Page column 73 ;