反应条件
1: tris-(dibenzylideneacetone)dipalladium(0); caesium carbonate; 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl / N,N-dimethyl-formamide / 18 h / 80 °C
2: water; tin(ll) chloride / methanol; ethyl acetate / 18 h / Reflux
View Scheme
参考文献
Burgeson, James R.; Moore, Amy L.; Boutilier, Jordan K.; Cerruti, Natasha R.; Gharaibeh, Dima N.; Lovejoy, Candace E.; Amberg, Sean M.; Hruby, Dennis E.; Tyavanagimatt, Shanthakumar R.; Allen III, Robert D.; Dai, Dongcheng
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 13 p. 4263 - 4272