6-甲氧基-2,3,4,5-四氢-1H-苯并[b]氮杂卓盐酸盐合成路线 (共 1 条)
反应条件
1: With diisobutylaluminium hydride in hexane; dichloromethane
T=0°C; 2 h;
2: With water; NAF in hexane; dichloromethane
2 h; Product distribution / selectivity;
参考文献
Szewczyk, Jerzy Ryszard; Donaldson, Kelly H.
Patent: US2006/3991 A1, 2006 ;
Location in patent: Page/Page column 19 ;
US 20060003991 A1