1: sodium hydroxide / 2 h / 20 °C
2: neat (no solvent) / 1 h / 125 °C
3: hydrogen bromide / water / 24 h / 70 °C
4: triethylamine / dichloromethane / 0 - 20 °C
View Scheme
参考文献
Hofer, Sandra; Kratschmar, Denise V.; Schernthanner, Brigitte; Vuorinen, Anna; Schuster, Daniela; Odermatt, Alex; Easmon, Johnny
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 19 p. 5397 - 5400