反应条件
1.1: 90 percent / HBr; AcOH 2.1: 95 percent / (COCl)2 / CH2Cl2 3.1: Wang resin; Hunig's base / CH2Cl2 / 0 - 20 °C 3.2: CsF; Pd(PPh3)4 / 1,2-dimethoxy-ethane / 10 h / 95 °C 3.3: TFA / CH2Cl2 / 0.17 h / 20 °C View Scheme
参考文献
Juteau, Helene; Gareau, Yves; Labelle, Marc; Lamontagne, Sonia; Tremblay, Nathalie; Carriere, Marie-Claude; Sawyer, Nicole; Denis, Danielle; Metters, Kathleen M.
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 5 p. 747 - 749