反应条件
1: 6-[5-(2-oxo-hexahydro-thieno[3,4-d]imidazol-4-yl)-pentanoylamino]-hexanoic acid With pyridine; dicyclohexyl-carbodiimide in N,N-dimethyl-formamide T=20°C; 0.0833333 h; 2: 1-hydroxy-pyrrolidine-2,5-dione in N,N-dimethyl-formamide 18 h;
参考文献
Wang, Tzu-Pin; Chiou, Yi-Jang; Chen, Yi; Wang, Eng-Chi; Hwang, Long-Chih; Chen, Bing-Hung; Chen, Yen-Hsu; Ko, Chun-Han
Bioconjugate Chemistry, 2010 , vol. 21, # 9 p. 1642 - 1655