反应条件
dicyclohexyl-carbodiimide in tetrahydrofuran
T=21°C; Substitution; 5 h; educts dissolving in THF; DCC adding dropwise, stirring; dicyclohexylurea filtering off; concng., washing, drying on MgSO4;
参考文献
De Tullio, Pascal; Pirotte, Bernard; Neven, Philippe; Masereel, Bernard; Dewalque, Daniel; Diouf, Ousmane; Podona, Tchao; Caignard, Daniel; Renard, Pierre; Delarge, Jacques
Journal of Pharmacy and Pharmacology, 1997 , vol. 49, # 5 p. 463 - 471