1: With copper(l) iodide in DMF (N,N-dimethyl-formamide)
T=120°C; 40 h;
2: With sodium hydrogencarbonate in DMF (N,N-dimethyl-formamide); dichloromethane; water
T=20°C;
参考文献
GLAXO GROUP LIMITED
Patent: WO2005/26125 A1, 2005 ;
Location in patent: Page/Page column 20 ;
WO 2005/026125 A1