1: 59 percent / rac-BINAP; Pd(OAc)2; Cs2CO3 / toluene / 20 h / Heating 2: 1.5 h / 105 °C View Scheme
参考文献
Kenny, Jane R.; Maggs, James L.; Meng, Xiaoli; Sinnott, Deborah; Clarke, Stephen E.; Park, B. Kevin; Stachulski, Andrew V.
Journal of Medicinal Chemistry, 2004 , vol. 47, # 11 p. 2816 - 2825
1: 59 percent / rac-BINAP; Pd(OAc)2; Cs2CO3 / toluene / 20 h / Heating 2: 1.5 h / 105 °C 3: 0.35 g / AlCl3 / 2 h / 150 °C 4: 38 percent / AlCl3 / 4 h / 200 - 210 °C View Scheme
参考文献
Kenny, Jane R.; Maggs, James L.; Meng, Xiaoli; Sinnott, Deborah; Clarke, Stephen E.; Park, B. Kevin; Stachulski, Andrew V.
Journal of Medicinal Chemistry, 2004 , vol. 47, # 11 p. 2816 - 2825
Wolfe, James F.; Rathman, Terry L.; Sleevi, Mark C.; Campbell, James A.; Greenwood, Thomas D.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 1 p. 161 - 166