反应条件
1: 1.) PBr3, 2.) HBr (g) / 1.) CH3Cl, 60 deg C, 30 min, 2.) CH3Cl, ether
2: 10 percent / tetrabutylammonium chloride / acetonitrile / 72 h / Ambient temperature
View Scheme
参考文献
Novella Romanelli; Teodori; Scapecchi; Dei; Budriesi; Chiarini
Farmaco, 1991 , vol. 46, # 10 p. 1121 - 1138