4,6-二氯-2-(氯甲基)喹唑啉合成路线 (共 2 条)
反应条件
hydrogenchloride in 1,4-dioxane
T=0 - 20°C;
参考文献
F. HOFFMANN-LA ROCHE AG; HOFFMANN-LA ROCHE INC.; FLOHR, Alexander; GROEBKE ZBINDEN, Katrin; KOERNER, Matthias; LERNER, Christian
Patent: WO2013/178569 A1, 2013 ;
Location in patent: Page/Page column 39-40 ;
参考文献
Hoffmann-La Roche Inc.
Patent: US5387585 A1, 1995 ;
US 5387585 A