反应条件
O-(benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate; triethylamine in N,N-dimethyl-formamide
T=20°C; 16 h;
参考文献
Zhao, Hongyu; Serby, Michael D.; Xin, Zhili; Szczepankiewicz, Bruce G.; Liu, Mei; Kosogof, Christi; Liu, Bo; Nelson, Lissa T. J.; Johnson, Eric F.; Wang, Sanyi; Pederson, Terry; Gum, Rebecca J.; Clampit, Jill E.; Haasch, Deanna L.; Abad-Zapatero, Cele; Fry, Elizabeth H.; Rondinone, Cristina; Trevillyan, James M.; Sham, Hing L.; Liu, Gang
Journal of Medicinal Chemistry, 2006 , vol. 49, # 15 p. 4455 - 4458