反应条件
1: 2-amino-phenol With calcium carbonate in 1,4-dioxane
T=70°C; 1.33333 h;
2: N-morpholinecarbonyl chloride in 1,4-dioxane
T=70 - 80°C; 0.75 h;
参考文献
Hernandez-Olmos, Victor; Abdelrahman, Aliaa; El-Tayeb, Ali; Freudendahl, Diana; Weinhausen, Stephanie; Mueller, Christa E.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 22 p. 9576 - 9588