1: With magnesium in tetrahydrofuran T=20°C; 2 h; 2: With N,N-dimethyl-formamide in tetrahydrofuran T=0°C; 2 h; 3: With ammonia; iodine in tetrahydrofuran; water T=20°C; 2 h;
titanium(IV) isopropylate; tributylphosphine in dichloromethane T=20°C; 15 h;
参考文献
Palmelund, Anders; Myers, Eddie L.; Tai, Lik Ren; Tisserand, Steve; Butts, Craig P.; Aggarwal, Varinder K.
Chemical Communications, 2007 , # 40 p. 4128 - 4130