2-乙基-4-(4-甲基哌嗪-1-基)-10h-苯并[b]噻吩并[2,3-e][1,4]二氮杂卓合成路线 (共 2 条)
反应条件
titanium tetrachloride in various solvent(s)
T=120°C; 2 h;
参考文献
Chakrabarti, Jiban K.; Horsman, Linda; Hotten, Terrence M.; Pullar, Ian A.; Tupper, David E.
Journal of Medicinal Chemistry, 1980 , vol. 23, # 8 p. 878 - 884
参考文献
IVAX CORPORATION
Patent: WO2003/104239 A1, 2003 ;
Location in patent: Page 8-10 ;
WO 03/104239 A1