反应条件
1: pyridine-2-carboxylic acid With benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; N-ethyl-N,N-diisopropylamine in 1,4-dioxane
T=20°C;
2: 3-trifluoromethyl-aniline in 1,4-dioxane
T=50°C;
参考文献
Engers, Darren W.; Niswender, Colleen M.; Weaver, C. David; Jadhav, Satyawan; Menon, Usha N.; Zamorano, Rocio; Conn, P. Jeffrey; Lindsley, Craig W.; Hopkins, Corey R.
Journal of Medicinal Chemistry, 2009 , vol. 52, # 14 p. 4115 - 4118