反应条件
thionyl chloride in N,N,N',N',N'',N''-hexamethylphosphoric triamide
T=-5°C; 0.166667 h;
参考文献
Hirai, Kentaro; Ishiba, Teruyuki; Sugimoto, Hirohiko; Fujishita, Toshio; Tsukinoki, Yuji; Hirose, Katsumi
Journal of Medicinal Chemistry, 1981 , vol. 24, # 1 p. 20 - 27