反应条件
1: triethylamine / dichloromethane / 0 - 20 °C
2: palladium diacetate; tris-(o-tolyl)phosphine; caesium carbonate; 2,2,2-trimethylacetic acid / 1-methyl-pyrrolidin-2-one / 48 h / 140 °C / |Schlenk technique
View Scheme
参考文献
Yan, Jia-Xuan; Li, Hu; Liu, Xiang-Wei; Shi, Jiang-Ling; Wang, Xin; Shi, Zhang-Jie
Angewandte Chemie - International Edition, 2014 , vol. 53, # 19 p. 4945 - 4949