反应条件
1: 3-bromo-4-methoxy-1-(triisopropylsilyl)-1H-indole With tert.-butyl lithium in tetrahydrofuran; pentane 0.25 h; Inert atmosphere; 2: 2-isopropoxy-4,4,5,5-tetramethyl-1,3,2-dioxaborolane in tetrahydrofuran; pentane T=-78°C; 1 h; Inert atmosphere;
参考文献
Lebar, Matthew D.; Hahn, Kristopher N.; Mutka, Tina; Maignan, Patrick; McClintock, James B.; Amsler, Charles D.; Van Olphen, Alberto; Kyle, Dennis E.; Baker, Bill J.
Bioorganic and Medicinal Chemistry, 2011 , vol. 19, # 19 p. 5756 - 5762