4-甲磺酰氨苯基硼酸频那醇酯合成路线 (共 2 条)
反应条件
4-methyl-morpholine in dichloromethane T=0 - 20°C; 2 h;
参考文献
SUGEN, INC.
Patent: WO2004/76412 A2, 2004 ;
Location in patent: Page 104 ;
WO 2004/076412 A2
反应条件
(1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium acetate in dichloromethane; N,N-dimethyl acetamide T=80°C;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 5 p. 1724 - 1727