1: With trans-N,N'-dimethylcyclohexane-1,2-diamine; 1,1,1,3,3,3-hexamethyl-disilazane; sodium iodide; copper(l) iodide in 1,4-dioxane T=110°C; 23 h; 2: With hydrogenchloride; water in 1,4-dioxane T=20°C;
参考文献
MASSACHUSETTS INSTITUTE OF TECHNOLOGY
Patent: WO2004/13094 A2, 2004 ;
Location in patent: Page 44 ;