Sellarajah, Shane; Lekishvili, Tamuna; Bowring, Claire; Thompsett, Andrew R.; Rudyk, Helene; Birkett, Christopher R.; Brown, David R.; Gilbert, Ian H.
Journal of Medicinal Chemistry, 2004 , vol. 47, # 22 p. 5515 - 5534
1: With triethylamine in tetrahydrofuran
T=0 - 20°C; 2 h;
2: With lithium aluminium tetrahydride in diethyl ether
T=0 - 20°C; 5 h;
3: With hydrogenchloride; 4-methylmorpholine N-oxide; tetrapropylammonium perruthennate
more than 3 stages;
参考文献
Genecare Research Institute Co., Ltd
Patent: EP1900728 A1, 2008 ;
Location in patent: Page/Page column 167 ;
