反应条件
1: With methanesulfonic acid in methanol T=80°C; Reflux; 2: With 4-(N,N-dimethlyamino)pyridine; acetic anhydride; triethylamine in dichloromethane T=50°C; 3: With water; potassium hydroxide in methanol T=50°C; 2 h;
参考文献
Kamino, Shinichiro; Kawamae, Yuko; Ijyuin, Megumi; Takada, Shingo; Yamaguchi, Takako; Doi, Mitsunobu; Fujita, Yoshikazu
Chemical and Pharmaceutical Bulletin, 2009 , vol. 57, # 12 p. 1405 - 1408