反应条件
EDC monohydrochloride; benzotriazol-1-ol; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide
T=20°C; 12 h;
参考文献
ENDO PHARMACEUTICALS INC.; SMITH, Roger, Astbury; THOMPSON, Scott, Kevin; HOSAHALLI, Subramanya; BEJUGAM, Mallesham; NANDURI, Srinivas; PANIGRAHI, Sunil, Kumar; MAHALINGAM, Natarajan
Patent: WO2012/58671 A1, 2012 ;
Location in patent: Page/Page column 74-75 ;