4-(3-氟苯基)-1,3-恶唑合成路线 (共 1 条)
反应条件
1: sodium formate; 1-(3-fluoro-phenyl)-ethanone in DMF (N,N-dimethyl-formamide)
T=20°C; 24 h;
2: ammonium acetate With acetic acid
1.5 h; Heating / reflux;
参考文献
Pfizer Inc.
Patent: US2003/225056 A1, 2003 ;
Location in patent: Page 46 ;