1: With N-bromosuccinmide; dibenzoyl peroxide in tetrachloromethane 36 h; 2: With N-ethyl-N,N-diisopropylamine; phosphonic acid diethyl ester in tetrahydrofuran T=20°C; 48 h; Further stages.;
参考文献
Charrier, Cedric; Roche, Joelle; Gesson, Jean-Pierre; Bertrand, Philippe
Bioorganic and Medicinal Chemistry Letters, 2007 , vol. 17, # 22 p. 6142 - 6146