反应条件
hydrogenchloride; 3 A molecular sieve; sodium cyanoborohydride
1.) EtOH, room temperature, 1 h, 2.) EtOH, room temperature, 3.) Et2O, AcOEt, room temperature; Yield given. Multistep reaction;
参考文献
Saito; Matsui; Fukushima; Watanabe; Waga; Kajiwara; Shirota; Iijima; Kitabatake
Arzneimittel-Forschung/Drug Research, 1989 , vol. 39, # 12 p. 1558 - 1561