反应条件
1: trifluoroacetic acid / dichloromethane 2: sodium hydride / dimethyl sulfoxide / 20 °C 3: ammonium formate / palladium on carbon / methanol 4: triethylamine / 4-(N,N-dimethlyamino)pyridine View Scheme
参考文献
MITHRIDION, INC.; ABRAHAM, Brent, D.; COPP, Richard, R.; FARNHAM, James, G.; HANSON, Seth, A.; HENDRICKSON, Michael, L.; OCKULY, Jeffrey, C.; TWOSE, Trevor, M.; VERDONE, Melinda, L.
Patent: WO2012/33956 A1, 2012 ;
WO 2012/033956 A1