反应条件
1: benzene-1,4-diol / benzene / 96 h / 180 °C
2: H2 / Pd-C / ethyl acetate
3: (i) CuBr2, AcOEt, CHCl3, (ii) Li2CO3, LiBr, DMF
View Scheme
参考文献
Cashin; Fairhurst; Horwell; et al.
European Journal of Medicinal Chemistry, 1978 , vol. 13, # 6 p. 495 - 501