1-(4-氟苯基)-1,3-二氢-1-[3-(甲基氨基)丙基]异苯并呋喃-5-甲腈合成路线 (共 1 条)
反应条件
1: With formic acid in chloroform 8 h; Heating / reflux; 2: With ammonia in chloroform; water T=20°C; pH=8 - 9;
参考文献
WOCKHARDT LIMITED; JAWEED MUKARRAM, Siddiqui, Mohammed; BHARGAV, Krishnaji, Upadhye; MISHRA, Krishna, Gopalji; FAROOQUI, Mohammed, Ismail
Patent: WO2005/42473 A1, 2005 ;
Location in patent: Page/Page column 11 ;