1: 2-propanethiol With sodium hydride in tetrahydrofuran
T=50°C; 1 h;
2: 3-bromopyridine-2-carbonitrile in tetrahydrofuran
T=50°C; 1.5 h; Reflux;
参考文献
LG LIFE SCIENCES LTD.; AHN, Sei Chang; KIM, Sook Hee; LEE, Ju Young; YOON, Joo Yong; YOON, Man Young
Patent: WO2014/10990 A1, 2014 ;
Location in patent: Paragraph 182; 183; 184 ;