反应条件
1: 5,6-diamino-1-butyl-3-(3-fluoro-benzyl)-1H-pyrimidine-2,4-dione With 1H-imidazole; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride
2: N-acetyl-4-aminophenyl-acetic acid With 4-(N,N-dimethlyamino)pyridine in N,N-dimethyl-formamide
参考文献
Foley, Louise H.; Wang, Ping; Dunten, Pete; Ramsey, Gwendolyn; Gubler, Mary-Lou; Wertheimer, Stanley J.
Bioorganic and Medicinal Chemistry Letters, 2003 , vol. 13, # 20 p. 3607 - 3610