反应条件
1: 5-(2-methoxyphenoxy)-2-(pyrimidin-2-yl)tetrahydropyrimidine-4,6-dione With trichlorophosphate in toluene 0.5 h; 2: 4-tert-Butylphenylsulphonylamine With sodium carbonate in N,N-dimethyl-formamide T=110 - 115°C;
参考文献
CADILA PHARMACEUTICALS LTD; MODI, Rajiv Indravadan; GUDAPARTHI, Omprakash; CHOWDHARY, Anil Shankar; KUMAR, Neeraj; GAVALE, Sharad Natthu; SONI, Sanjay Kanhaiyalal; PATEL, Nilesh Govind; PANDIT, Unnat Priyavadan
Patent: WO2013/186706 A1, 2013 ;
Location in patent: Page/Page column 8 ;