反应条件
1: With pyridine; ethyl orthosilicate; pyridinium p-toluenesulfonate T=20°C; 24 h; 2: With tetrakis(triphenylphosphine) palladium(0); N,N-dicyclohexylmethylamine T=160°C; 0.333333 h; Microwave irradiation;
参考文献
Engelhardt, Harald; De Esch, Iwan J.P.; Kuhn, Daniel; Smits, Rogier A.; Zuiderveld, Obbe P.; Dobler, Julia; Mayer, Moriz; Lips, Sebastian; Arnhof, Heribert; Scharn, Dirk; Haaksma, Eric E.J.; Leurs, Rob
European Journal of Medicinal Chemistry, 2012 , vol. 54, p. 660 - 668