1: With borane in tetrahydrofuran T=90°C; 14.3333 h; 2: With water in tetrahydrofuran 0.5 h; 3: With hydrogenchloride; water in tetrahydrofuran pH=2; 5 h;
参考文献
SMITHKLINE BEECHAM CORPORATION
Patent: WO2003/74495 A1, 2003 ;
Location in patent: Page/Page column 64 ;
WO 03/074495 A1