1: 57 percent / tert-butyl nitrite; diidodomethane / acetonitrile / 2.5 h / 80 °C 2: 48 percent / aq. NaOH / propan-2-ol / 72 h / 20 °C View Scheme
参考文献
Kim, Hak Sung; Ohno, Michihiro; Xu, Bin; Kim, Hea Ok; Choi, Yongseok; Ji, Xiao D.; Maddileti, Savitri; Marquez, Victor E.; Harden, T. Kendall; Jacobson, Kenneth A.
Journal of Medicinal Chemistry, 2003 , vol. 46, # 23 p. 4974 - 4987