7-[[4-[(4-氯苯基)甲氧基]苯基]磺酰基]-2,3,4,5-四氢-8-甲氧基-3-甲基-1H-3-苯并氮杂卓合成路线 (共 1 条)
反应条件
1: 4-chloro-1-hydroxymethyl-benzene With potassium tert-butylate in tetrahydrofuran
T=25°C; 0.166667 h;
2: 7-(4-fluoro-benzenesulfonyl)-8-methoxy-3-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine in tetrahydrofuran
T=25°C; 1.75 h;
参考文献
GLAXO GROUP LIMITED
Patent: WO2005/51916 A1, 2005 ;
Location in patent: Page/Page column 7; 27 ;
WO 2005/051916 A1