1: With water; sodium hydroxide in methanol
T=20°C; Inert atmosphere;
2: With hydrogenchloride in dichloromethane; water
参考文献
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA; NATIONAL INSTITUTES OF HEALTH; COHEN, Seth M.; AGRAWAL, Arpita; DESOTO, Jamie; POMMIER, Yves; MADDALI, Kasthuraiah
Patent: WO2012/106534 A2, 2012 ;
Location in patent: Page/Page column 67 ;
WO 2012/106534 A2