反应条件
1: in N,N-dimethyl-formamide
T=85°C; 6 h;
2: With copper(l) iodide; caesium carbonate; L-proline in N,N-dimethyl-formamide
T=80 - 85°C; 6 h;
参考文献
Maity, Arindam; Mondal, Shyamal; Paira, Rupankar; Hazra, Abhijit; Naskar, Subhendu; Sahu, Krishnendu B.; Saha, Pritam; Banerjee, Sukdeb; Mondal, Nirup B.
Tetrahedron Letters, 2011 , vol. 52, # 23 p. 3033 - 3037