反应条件
benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=20°C; 12 h; Inert atmosphere;
参考文献
Greguric, Ivan; Taylor, Stephen R.; Denoyer, Delphine; Ballantyne, Patrice; Berghofer, Paula; Roselt, Peter; Pham, Tien Q.; Mattner, Filomena; Bourdier, Thomas; Neels, Oliver C.; Dorow, Donna S.; Loc'h, Christian; Hicks, Rodney J.; Katsifis, Andrew
Journal of Medicinal Chemistry, 2009 , vol. 52, # 17 p. 5299 - 5302