1: 97 percent / TEA; HOBt; EDCl / dimethylformamide / 5 h / 20 °C 2: 94 percent / TEA / methanol / 24 h / 60 °C View Scheme
参考文献
Park Choo, Hea-Young; Kim, Mihyun; Lee, Sang Kook; Woong Kim, Sang; Kwon Chung, In
Bioorganic and Medicinal Chemistry, 2002 , vol. 10, # 3 p. 517 - 523