反应条件
1: SOCl2 / CHCl3 / Heating
2: toluene / Ambient temperature
3: 1.) t-BuLi / 1.) THF, -78 deg C, 15 min, 2.) THF, from -78 to -65 deg C, 4 h
View Scheme
参考文献
Pettit, George R.; Toki, Brian; Herald, Delbert L.; Verdier-Pinard, Pascal; Boyd, Michael R.; Hamel, Ernest; Pettit, Robin K.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 10 p. 1688 - 1695