1H-吡唑并[3,4-c]吡啶-5-甲腈合成路线 (共 1 条)
反应条件
tetrakis(triphenylphosphine) palladium(0) in N,N-dimethyl-formamide
T=180°C; 0.5 h; Inert atmosphere;
参考文献
ALLERGAN, INC.; CARLING, William R.; MARTOS, Jose L.; KANGASMETSA, Jussi J.; WANG, Jenny W.; WOODWARD, David F.
Patent: WO2013/96496 A2, 2013 ;
Location in patent: Page/Page column 112 ;