1: hydrogenchloride / ethylene glycol dimethyl ether; water / 4 h / Reflux 2: palladium 10 on activated carbon; hydrogen / methanol / 72 h View Scheme
参考文献
Conway, Richard J.; Valant, Celine; Christopoulos, Arthur; Robertson, Alan D.; Capuano, Ben; Crosby, Ian T.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 7 p. 2560 - 2564