反应条件
1.1: 1,1'-carbonyldiimidazole / tetrahydrofuran / 2 h / 20 °C 1.2: 20 °C 2.1: dihydrogen peroxide; acetic acid / methanol; water / 24 h / 40 °C 3.1: lithium aluminium tetrahydride; sulfuric acid / tetrahydrofuran / 2 h / 20 °C View Scheme
参考文献
Cao, Jianjing; Prisinzano, Thomas E.; Okunola, Oluyomi M.; Kopajtic, Theresa; Shook, Matthew; Katz, Jonathan L.; Newman, Amy Hauck
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 1 p. 48 - 52