4-溴-2-氟-N-羟基-苯甲脒合成路线 (共 2 条)
反应条件
sodium hydride in tetrahydrofuran
T=60°C; 15 h; Molecular sieveHeating / reflux;
参考文献
RANBAXY LABORATORIES LIMITED
Patent: WO2006/38100 A1, 2006 ;
Location in patent: Page/Page column 75 ;
反应条件
in pyridine
T=20°C; 17 h; Heating / reflux;
参考文献
PFIZER INC.
Patent: WO2004/74270 A2, 2004 ;
Location in patent: Page 50 ;